1020920-65-3Relevant academic research and scientific papers
Synthesis and herbicidal activity of N-aryl-2-heteroaryloxy-N-isopropyl acetamide
Ye, Qing,Zhu, Xiao-Bo,Gu, Kai,Ni, Xiao-Quan,Gao, Jian-Rong,Wei-Rong, Miao
, p. 6931 - 6934 (2013/07/26)
A series of novel N-aryl-2-heteroaryloxy-N-isoproylacetamide derivatives were synthesized by multi-step reactions. Their structures were characterized by 1H NMR, MS and elemental analyses. The target compounds were evaluated for their herbicidal activities against Echinochloa crusgalli, Digitaria sanguinalis Scop., Abutilon theophrasti, Setaria viridis, Zinnia elegans and Acalypha australis. The results indicated that some of the title compounds displayed excellent herbicidal activities.
CCK or gastrin modulating benzo ?b!?1,4! diazepines derivatives
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, (2008/06/13)
Benzo?b!?1,4!diazepine compounds of formula (I), where R1 is selected from C1 C6 alkyl, C3 -C6 cycloalkyl, phenyl, or substituted phenyl; R2 is selected from C3 -C6 alkyl, C3 C6 cycloalkyl, C3 -C6 alkenyl, benzyl, phenylC1 -C3 alkyl of substituted phenyl; or NR1 R2 together form 1,2,3,4-tetrahydroquinoline or benzazepine, mono-, di-, or trisubstituted independently with C1-6 alkyl C1-6 alkoxy or halogen substituents; p is an integer 0 or 1; q is an integer 0 or 1; r is an integer 0 or 1; t is an integer 0 or 1, provided that when r is 0 then t is 0; R3, R5, and R6 are independently hydrogen or C1-6 alkyl; R4 is C1-6 alkyl or C1-6 alkenyl; R7 is selected from the group consisting of hydrogen, C1-6 alkyl, C1-6 cycloalkyl, C1-6 alkenyl, phenyl, substituted phenyl, napthyl, heteroaryl, substituted heteroaryl, bicycloheteroaryl or substituted bicycloheteroaryl; or NR6 R7 together form a saturated 5,6, or 7 membered ring optionally interrupted by 1,2,3 or 4 N, S or O heteroatoms, with the proviso that any two O or S atoms are not bonded to each other, m is an integer selected from the group of 0, 1, 2, 3 or 4; R8 and R9 are selected from a variety of substituents; Z is hydrogen or halogen; novel intermediates, a pharmaceutical composition for treating obesity, gall bladder stasis, disorders of pancreatic secretion, methods for such treatment and processes for preparing compounds of formula (I).
