1027150-97-5Relevant academic research and scientific papers
3-[2-(N-phenylacetamide)]-1,5-benzodiazepines: Orally active, binding selective CCK-A agonists
Willson, Timothy M.,Henke, Brad R.,Momtahen, Tanya M.,Myers, Peter L.,Sugg, Elizabeth E.,Unwalla, Rayomand J.,Croom, Dallas K.,Dougherty, Robert W.,Grizzle, Mary K.,Johnson, Michael F.,Queen, Kennedy L.,Rimele, Thomas J.,Yingling, Jeffrey D.,James, Michael K.
, p. 3030 - 3034 (2007/10/03)
A series of modifications were made to the C-3 substituent of the 1,5- benzodiazepine CCK-A agonist 1. Replacement of the inner urea NH and addition of a methyl group to generate a C-3 quaternary carbon resulted in acetamide 6, which showed CCK-A receptor
