1027982-33-7Relevant academic research and scientific papers
Inhibition of stromelysin-1 (MMP-3) by P1'-biphenylylethyl carboxyalkyl dipeptides
Esser, Craig K.,Bugianesi, Robert L.,Caldwell, Charles G.,Chapman, Kevin T.,Durette, Philippe L.,Girotra, Narindar N.,Kopka, Ihor E.,Lanza, Thomas J.,Levorse, Dorothy A.,MacCoss, Malcolm,Owens, Karen A.,Ponpipom, Mitree M.,Simeone, Joseph P.,Harrison, Richard K.,Niedzwiecki, Lisa,Becker, Joseph W.,Marcy, Alice I.,Axel, Melinda G.,Christen, Amy J.,McDonnell, Joseph,Moore, Vernon L.,Olszewski, Julie M.,Saphos, Cheryl,Visco, Denise M.,Shen, Frank,Colletti, Adria,Krieter, Philip A.,Hagmann, William K.
, p. 1026 - 1040 (1997)
Carboxyalkyl peptides containing a biphenylylethyl group at the P1' position were found to be potent inhibitors of stromelysin-1 (MMP-3) and gelatinase A (MMP-2), in the range of 10-50 nM, but poor inhibitors of collagenase (MMP-1). Combination
