107036-26-0Relevant articles and documents
Estrogenic Affinity Labels: Synthesis, Irreversible Receptor Binding, and Bioactivity of Aziridine-Substituted Hexestrol Derivatives
Zablocki, Jeffery A.,Katzenellenbogen, John A.,Carlson, Kathryn E.,Norman, M. J.,Katzenellenbogen, Benita S.
, p. 829 - 838 (2007/10/02)
To develop an affinity label for the estrogen receptor that would be an estrogen agonist, rather than antagonist, we prepared several aziridine derivatives of the potent nonsteroidal estrogen hexestrol (3R*,4S*)-3,4-bis(4-hydroxyphen