1144044-87-0Relevant academic research and scientific papers
Synthesis and SAR studies of trisubstituted purinones as potent and selective adenosine A2A receptor antagonists
Shao, Yuefei,Cole, Andrew G.,Brescia, Marc-Raleigh,Qin, Lan-Ying,Duo, Jingqi,Stauffer, Tara M.,Rokosz, Laura L.,McGuinness, Brian F.,Henderson, Ian
scheme or table, p. 1399 - 1402 (2009/10/15)
A series of trisubstituted purinones was synthesized and evaluated as A2A receptor antagonists. The A2A structure-activity relationships at the three substituted positions were studied and selectivity against the A1 recept
TRIAZOLOPYRIMIDINE DERIVATIVES AS GLYCOGEN SYNTHASE KINASE 3 INHIBITORS
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Page/Page column 37, (2008/06/13)
This invention concerns a compound of formula (I), a N-oxide, a pharmaceutically acceptable addition salt, a quaternary amine and a stereochemically isomeric form thereof, wherein ring A represents phenyl, pyridyl, pyrimidinyl, pyridazinyl or pyrazinyl; R
