118602-96-3Relevant academic research and scientific papers
7-(MORPHOLIN-4-YL)PYRAZOLE[1,5-A]PYRIMIDINE DERIVATIVES WHICH ARE USEFUL FOR THE TREATMENT OF IMMUNE OR INFLAMMATORY DISEASES OR CANCER
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, (2017/07/31)
A compound of the general formula (I) wherein Y represents -CH2- or >C=0; R1 is selected from the group consisting of A1, A2 and A3; R2 represents dioxothiomorpholino moiety B1, piperazinyl moiety B2, azetidinyl moiety B3, or piperidinyl moiety B4; R3 is selected from the group consisting of H, halogen, and C1 -C4 alkyl; R4 is selected from the group consisting of C1 -C4 alkyl, C3-C4- cycloalkyl, C1 -C4 alkyl substituted with C1 -C4 alkoxy, and CHF2, and their pharmaceutically acceptable salts. Pharmaceutical compositions comprising said compounds and their use in the treatment of diseases of immune system, inflammatory diseases and cancer.
HERBICIDAL ISOXAZOLO[5,4-B]PYRIDINES
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Page/Page column 47, (2013/07/25)
The invention relates to isoxazolo[5,4-b]pyridine compounds of formula (I), to the agriculturally useful salts of isoxazolo[5,4-b]pyridine compounds of formula (I), and to their use as herbicides.
HETEROCYCLIC COMPOUNDS AS INHIBITORS OF CXCR2
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Page/Page column 31, (2009/10/21)
The present invention relates to compounds of formula (I) wherein R1, R2, X, Y and Z are as defined in the specification.
4,7-dihydroisothiazolo(5,4-b)pyridine derivatives and cardiovascular treating agents containing said derivatives
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, (2008/06/13)
A 4,7-dihydroisothiazole[5,4-b]pyridine derivative represented by the general formula STR1 wherein R1 represents an alkyl group which may be substituted, R2 represents a hydrogen atom, a hydroxyl group, a benzyloxy group, a lower alk
