119003-97-3Relevant academic research and scientific papers
Studies on the chemistry of O,N- and S,N-containing heterocycles. 3 [1]. Synthesis of 1,5-benzothiazepines with potential CNS activity
Bartsch,Erker
, p. 1151 - 1154 (1988)
The synthesis of a series of novel triazolo[3,4-d][1,5]benzothiazepines 6 and 7, obtained from the activated 1,5-benzothiazepine derivatives 3 and carbohydrazides 4,is described. Under mild reaction conditions some intermediates 5 can be isolated.
Studies of annelated 1,4-benzothiazines and 1,5-benzothiazepines. VII. Synthesis and inhibition of benzodiazepine receptor binding of some 4,5-dihydro-tetrazolo[5,1-d]-1,5-benzothiazepines and 5-phenyl-s-triazolo[3,4-d]-1,5-benzothiazepines
Ambrogi,Grandolini,Perioli,Giusti,Lucacchini,Martini
, p. 665 - 676 (2007/10/02)
The 4,5-dihydro-tetrazolo[5,1-d]-1,5-benzothiazepines 3a-k and the 5-phenyl-s-triazolo[3,4-d]-1,5-benzothiazepines 6a-f and 11a-c have been prepared and tested for their ability to displace [H] flunitrazepam binding from bovine brain membranes. Some of th
