1198312-18-3Relevant academic research and scientific papers
Benzenesulfonyl-Asymmetric Ureas and Medical Uses Thereof
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Paragraph 0198; 0206, (2017/10/10)
Benzenesulfonyl-asymmetric ureas are provided for the treatment of conditions modulated by the ghrelin receptor.
Discovery and optimization of novel 4-[(aminocarbonyl)amino]-N-[4-(2-aminoethyl)phenyl]benzenesulfonamide ghrelin receptor antagonists
Pasternak, Alexander,Goble, Stephen D.,deJesus, Reynalda K.,Hreniuk, Donna L.,Chung, Christine C.,Tota, Michael R.,Mazur, Paul,Feighner, Scott D.,Howard, Andrew D.,Mills, Sander G.,Yang, Lihu
scheme or table, p. 6237 - 6240 (2010/07/02)
This Letter describes optimization of ghrelin receptor antagonists and inverse agonists starting from a screening hit.
