120740-07-0Relevant academic research and scientific papers
Thiazolyl anabasine compound as well as preparation method and application thereof
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Paragraph 0023; 0025; 0027, (2018/09/21)
The invention discloses a thiazolyl anabasine compound as well as a preparation method and application thereof. The structure formula of the thiazolyl anabasine compound is shown as formula I, wherein R1 is hydrogen, methyl or ethyl; R2 is hydrogen, methyl, 2-chlorine-5-thiazole methyl or 6-chlorine-3-picolyl; 2-chlorine-5-chloromethyl thiazole reacts with ethylamine, so as to generate 2-chlorine-5-ethylamine methyl thiazole; and then, 1,1-dichloro nitro ethylene or 1,1,1-trichloronitroethane, 2-chlorine-5-ethylamine methyl thiazole and compound R1NH2R2 react under the existence of alkali, thereby generating the thiazolyl anabasine compound. The thiazolyl anabasine compound disclosed by the invention can be independently prepared into an insecticide and also can be mixed with other pesticides for preparing the insecticide. The thiazolyl anabasine compound disclosed by the invention has the advantages of high insecticidal activity, low toxicity, wide insecticidal spectrum, and the like, and has obvious insecticidal effect for plant hoppers, aphids, and the like.
Substituted benzisothiazole compound and application
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Paragraph 0158; 0160; 0161; 0162, (2018/03/24)
The invention discloses a substituted benzisothiazole compound. R1 is cyan, hydroxyl, C1-C4 alkyl, cyclopropyl, cyanomethyl, methoxyl, ethyoxyl, acetyl, trifluoroacetyl, C1-C4 alkoxycarbonyl and methylsulfonyl or ethylsulfonyl, R2 is independently selected from hydrogen, halogen, cyan, methyl, methoxyl, trifluoromethyl and trifluoromethoxyl or difluoromethoxyl, n is 1, 2, 3 or 4, m is 1 or 2, and J is replaced thiazole, isothiazole or pyridine. The compound has excellent activity and good plant tolerance and environmental safety under low concentration and can inhibit or destroy various pathogenic fungi and bacteria generated by plants or soil and kill various insect pests and mites, and sterilization and insecticidal spectrums of the compound are widened. According to the preparation method, used raw materials are economical and easy to get, and the preparation method is high in yield and low in synthesis process cost and has good sterilization activity and pest and mite killing activity.
Thiazole Methylamino Pyridine Compounds and Preparation Method Therefor
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Paragraph 0060-0061, (2015/02/25)
Disclosed are thiazole methylamino pyridine compounds represented by the general formula (I) having fungicidal, insecticidal/acaricidal, and herbicidal activity, the preparation method thereof, the fungicidal, insecticidal/acaricidal, and herbicidal compositions containing the compounds of the present invention, and the use and the method for controlling fungi, insects/acari and weeds of the compounds of the present invention.
