1228019-06-4

Upstream product

• 59-23-4 D-Galactose 
• 98-88-4 benzoyl chloride 
• 93-97-0 benzoic acid anhydride 
• 10257-28-0 D-Galactose 

Downstream Products

• 1228019-07-5 1,2,3,6-tetra-O-benzoyl-4-fluoro-β-glucopyranoside 
• 69534-71-0 1,2,3,6-tetra-O-benzoyl-4-deoxy-α-L-threo-hex-4-enopyranose 
• 461025-92-3 2,3,6-tri-O-benzoyl-4-deoxy-4-fluoro-α-D-glucopyranosyl bromide 
• 1228019-10-0 C₃₅H₂₇F₃O₁₂S 
• 1228019-04-2 1-O-acetyl-2,3,6-tri-O-benzoyl-4-fluoro-4-deoxy-α-D-glucose 

Relevant academic research and scientific papers

Process development of selectively benzoylated and fluorinated glycosyl donors

Route selection, process development and large-scale preparation of selectively benzoylated and fluorinated d-glucopyranoses, required as glycosyl donors for the synthesis of the SGLT inhibitor SAR7226, are discussed.

INTERMEDIATES AND PROCESSES FOR THE PREPARATION OF FLUOROGLYCOSIDE DERIVATIVES

The present invention provides processes for producing (2S,3R,4R,5S,6R)-5-fluoro-6- hydroxymethyl-2-[4-(4-methoxy-benzyl)-5-trifluoromethyl-1H-pyrazol-3-yloxy]- tetrahydro-pyran-3,4-diol or a tautomer or hydrate thereof, of high purity and in a relatively