125033-98-9Relevant academic research and scientific papers
2-KETO AMIDE DERIVATIVES AS HIV ATTACHMENT INHIBITORS
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Page/Page column 67-68, (2014/10/15)
Compounds of Formula I, including pharmaceutically acceptable salts thereof: I useful as HIV attachment inhibitors.
Synthetic potentiality of α-amino nitrones as oxidizing reagent in the conversion of alkyl halides to aldehydes
Chakraborty, Bhaskar,Chhetri, Manjit Singh,Kafley, Saurav,Sharma, Prawin,Rai, Neelam
experimental part, p. 1399 - 1402 (2011/09/20)
α-Amino nitrones have been used successfully as an oxidizing reagent for the synthesis of aldehydes from various alkyl halides with an excellent yield. In addition, hydrolysis of the side product (imines) furnishes starting material amides which are recyclable along with corresponding amines.
A Convenient Synthesis of N-Substituted Formamidines by Desulfurization of the Corresponding Thioureas
Kashima, Choji,Shimizu, Masao,Eto, Takeshi,Omote, Yoshimori
, p. 3317 - 3319 (2007/10/02)
N,N'-Di- and N,N,N'-trisubstituted thioureas were easily desulfurized by Raney nickel to yield the corresponding formamidines, while N-monosubstituted thioureas gave N,N'-disubstituted formamidines.
Raney Nickel Desulphuration of 1-Substituted- and 1,3-Disubstituted-thioureas
Ali, M. Umar,Meshram, H. M.,Paranjpe, M. G.
, p. 666 - 669 (2007/10/02)
Certain 1-aryl-1,3-diaryl- and 1-aryl-3-tetra-O-acetyl-β-D-glucopyranosyl thioureas have been successfully desulphurated into the related mono- and 1,3-di-substituted formamidines with the help of Raney nickel catalyst.A few of them have been converted into the corresponding formamides also.Structure of the products have been established through usual chemical transformations, ir, nmr and mass spectral analysis.
