125224-63-7Relevant articles and documents
Preparation of 2,5-diazabicyclo[2.2.1]heptanes and intermediates
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, (2008/06/13)
(R,R)-2,5-Diazabicyclo[ 2.2.1]heptanes are prepared from a compound of the formula STR1 wherein X and R2 are as defined herein, by heating with tosylchloride in pyridine, reacting the formed compound of the formula STR2 with a C1 -C6 alkylamine or ammonia, and reducing or hydrolyzing the formed compound of the formula STR3 wherein R1 is hydrogen or C1 -C6 alkyl.
Synthesis of (1R,4R)- and (1S,4S)-2,5-diazabicyclo[2.2.1]heptanes and their N-substituted derivatives
Jordis,Sauter,Siddiqi,Kuenburg,Bhattacharya
, p. 925 - 930 (2007/10/02)
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