126800-12-2Relevant academic research and scientific papers
Multi-component reaction for the preparation of 1,5-disubstituted 1,2,3-triazoles by in-situ generation of azides and nickel-catalyzed azide-alkyne cycloaddition
Camberlein, Virgyl,Kraupner, Nicolas,Bou Karroum, Nour,Lipka, Emmanuelle,Deprez-Poulain, Rebecca,Deprez, Benoit,Bosc, Damien
supporting information, (2021/05/10)
An efficient one-pot procedure combining bromide conversion into azide followed by NiAAC for the preparation of 1,5-disubstituted 1,2,3-triazoles has been developed. This procedure prevents the use of isolated azides, which are insufficiently commercially
A tunable route to oxidative and eliminative [3+2] cycloadditions of organic azides with nitroolefins: CuO nanoparticles catalyzed synthesis of 1,2,3-triazoles under solvent-free condition
Gangaprasad,Paul Raj,Kiranmye,Sasikala,Karthikeyan,Kutti Rani,Elangovan
supporting information, p. 3105 - 3108 (2016/07/06)
A regioselective and tunable synthesis of 1,5-disubstituted 1,2,3-triazloles from oxidative and eliminative [3+2] cycloadditions of nitroolefins and organic azides under solvent-free condition in the presence and absence of commercially available CuO nano
A general metal-free route towards the synthesis of 1,2,3-triazoles from readily available primary amines and ketones
Thomas, Joice,Jana, Sampad,John, Jubi,Liekens, Sandra,Dehaen, Wim
supporting information, p. 2885 - 2888 (2016/02/19)
An unprecedented approach that enables the direct and selective preparation of 1,5-disubstituted 1,2,3-triazoles from abundantly available building blocks such as primary amines, enolizable ketones and 4-nitrophenyl azide as a renewable source of dinitrogen via an organocascade process has been developed. Furthermore, this efficient methodology also enables the synthesis of fully functionalized and fused N-substituted heterocycles.
Designing 2-aminoimidazole alkaloids analogs with anti-biofilm activities: Structure-activities relationships of polysubstituted triazoles
Linares,Bottzeck,Pereira,Praud-Tabaris,Blache
experimental part, p. 6751 - 6755 (2011/12/21)
In order to discover novel probes that may help in the investigation and the control of bacterial biofilms, we have designed a library of triazole-based analogs of 2-aminoimidazole marine alkaloids: naamine A and isonaamine A. Twenty-two compounds were sc
Dipolar Cycloaddition Reactions of Organic Azides with some Acetylenic Compounds
Abu-Orabi, Sultan T.,Atfah, M. Adnan,Jibril, Ibrahim,Mari'i, Fakhri M.,Ali, Amer Al-Sheikh
, p. 1461 - 1468 (2007/10/02)
Phenyl azide 1 and several substituted benzyl azides 2a-o underwent 1,3-dipolar cycloaddition reactions with dimethyl acrtylenedicarboxylate 3, phenylacetylene 4 and ethyl propiolate 5 to afford the triazoles 6-13.The reactions of these azides with ethyl
