129141-69-1Relevant articles and documents
5-Fluorouracil derivatives. XX. Synthesis and antitumor activity of 5'-O-unsaturated acyl-5-fluorouridines
Ozaki,Akiyama,Morita,Kumegawa,Nagase,Uehara,Hoshi
, p. 3164 - 3166 (1990)
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p-Methoxybenzyl as a New N3-Imide Protecting Group of 5-Fluorouridine and Its Application to the Synthesis of 5'-O-Acryloyl-5-fluorouridine
Akiyama, Takahiko,Kumegawa, Masahiro,Takesue, Yasuhiro,Nishimoto, Hiroyuki,Ozaki, Shoichiro
, p. 339 - 342 (2007/10/02)
5'-O-Acryloyl-5-fluorouridine was prepared by use of p-methoxybenzyl (PMB) group as a new N3-imide protecting group of 5-fluorouridine.A chemoselective method for protection has been developed by use of ethyldiisopropylamine as a base and depro