13515-76-9Relevant articles and documents
Synthesis of novel benzoxaborole-containing phenylalanine analogues
Li, Xianfeng,Plattner, Jacob J.,Hernandez, Vincent,Ding, Charles Z.,Wu, Wei,Yang, Yang,Xu, Musheng
, p. 4924 - 4926 (2011)
The synthesis of novel benzoxaborole-containing phenylalanine analogues 2 and 3 has been developed. The key steps involve the preparation of appropriate precursors from the readily available amino acids and the formation of benzoxaborole ring directly in
BENZOTHIAZEPINE COMPOUNDS AND THEIR USE AS BILE ACID MODULATORS
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Paragraph 0673-0675, (2020/08/20)
The invention relates to 1,5-benzothiazepine derivatives of formula (I). These compounds are bile acid modulators having apical sodium-dependent bile acid transporter (ASBT) and/or liver bile acid transport (LBAT) inhibitory activity. The invention also r
MACROCYCLIC COMPOUNDS AS PROTEASOME INHIBITORS
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Paragraph 0507, (2019/05/02)
The compounds of the present invention are represented by the following compounds having Formula I and Formula (I'): where the substituents R1, R2, R2', R3, R4, R5, R', R", X, Y, and Z are as defined herein and where the substituents R1, R2, R3, R4, R5, R', R", X, Y, and Z are as defined herein. These compounds are used in the treatment of bacterial infections, parasite infections, fungal infections, cancer, immunologic disorders, autoimmune disorders, neurodegenerative diseases and disorders, inflammatory disorders, or muscular dystrophy or for providing immunosuppression for transplanted organs or tissues.