13532-16-6Relevant articles and documents
Aminothiolation of α-Bromocinnamaldehydes to Access Imidazo[2,1-b]thiazoles by Incorporation of Two Distinct Photoinduced Processes
Chen, Ziren,Jin, Weiwei,Xia, Yu,Zhang, Yonghong,Xie, Mengwei,Ma, Shangchao,Liu, Chenjiang
supporting information, p. 8261 - 8266 (2020/11/02)
A visible-light-promoted metal-free catalytic system was developed to achieve the aminothiolation of α-bromocinnamaldehydes. This mechanistically novel approach allows the synthesis of diverse imidazo[2,1-b]thiazole derivatives in satisfactory yields at r
DMAP-Catalyzed C—N Bond Formation for Diverse Synthesis of Imidazo[1,2-a]pyrimidine and Pyrimido[1,2-a]benzimidazole Derivatives
Shang, Le-Le,Feng, Yun,Gao, Xing-Lian,Chen, Zi-Ren,Xia, Yu,Jin, Wei-Wei,Liu, Chen-Jiang
supporting information, p. 1595 - 1599 (2020/10/02)
A DMAP (2-dimethylaminopyridine)-catalyzed condensation reactions for the successful direct construction of pyrimido[1,2-a]benzimidazole or imidazo[1,2-a]pyrimidine has been developed. The method utilizes readily available α-bromocinnamaldehydes with 2-am
NHC-Catalyzed Enantioselective [3 + 3] Annulation to Construct 5,6-Dihydropyrimidin-4-ones
Meng, Di,Xie, Yangxi,Peng, Qiupeng,Wang, Jian
supporting information, p. 7635 - 7639 (2020/10/09)
The unprecedented enantioselective NHC-catalyzed [3 + 3] annulation of α-bromoenals with amidines via a dual C-N bond formation is described. The protocol allows a rapid preparation of 5,6-dihydropyrimidinones in acceptable yields with good enantioselectivities.