1364569-59-4Relevant articles and documents
Anti-tumor activity of new orally bioavailable 2-amino-5-(thiophen-2-yl) benzamide-series histone deacetylase inhibitors, possessing an aqueous soluble functional group as a surface recognition domain
Hirata, Yoshiyuki,Hirata, Masahiko,Kawaratani, Yasuyuki,Shibano, Makio,Taniguchi, Masahiko,Yasuda, Masahide,Ohmomo, Yoshiro,Nagaoka, Yasuo,Baba, Kimiye,Uesato, Shinichi
, p. 1926 - 1930 (2012)
New orally bioavailable 5-(thiophen-2-yl)-substituted 2-aminobenzamide- series histone deacetylase inhibitors were synthesized. These compounds possess a morpholine or piperadine-derived moiety as an aqueous soluble functional group. Among them, 8b, havin