1380424-00-9Relevant articles and documents
Incorporation of an acyclic alkynyl nucleoside analog into siRNA improves silencing activity and nuclease resistance
Ogata, Aya,Ueno, Yoshihito
, p. 2574 - 2578 (2015/06/02)
In order to improve the silencing activity and nuclease resistance of small interfering RNA (siRNA), we designed and synthesized an acyclic thymidine analog containing 4-pentyne-1,2-diol instead of d-ribofuranose. The incorporation of this analog into siR