140706-33-8Relevant articles and documents
Ultrasound-assisted 3-component reaction in acetic acid alone: Catalyst/promoter/ligand free synthesis of bioactive pyrazolo[1,5-a]pyrimidines
Suresha, Namburi,Durgaraoa, Bodapati Veera,Ratnakar,Kolli, Sunder Kumar,Ashfaq, Mohd Ashraf,Rao, Mandava V. Basaveswara,Pal, Manojit
, p. 1176 - 1183 (2017/11/14)
Background: Acetic acid alone when employed as a solvent under ultrasound irradiation has been found to be effective for the three-component reaction involving ethyl-5- A mino-1H-pyrazole-4-carboxylate, aromatic aldehydes and terminal alkynes in the prese
Synthesis and structure-activity relationship of tetrahydropyrazolopyrimidine derivatives - A novel structural class of potent calcium-sensing receptor antagonists
Yoshida, Masato,Mori, Akira,Inaba, Atsuhiro,Oka, Masahiro,Makino, Haruhiko,Yamaguchi, Masashi,Fujita, Hisashi,Kawamoto, Tomohiro,Goto, Mika,Kimura, Hiroyuki,Baba, Atsuo,Yasuma, Tsuneo
experimental part, p. 8501 - 8511 (2011/02/23)
A series of novel tetrahydropyrazolopyrimidine derivatives containing an adamantyl group were synthesized and evaluated as potential calcium-sensing receptor (CaSR) antagonists. After chemical modification of 9a, which was identified as a hit compound in