144075-70-7

Upstream product

• 134210-24-5 methyl (4S,5S,2E)-5-amino-N-<(tert-butyloxy)carbonyl>-4-hydroxy-6-phenyl-2-hexanoate 
• 256463-36-2 methyl (2S,3S)-3-benzyl-1-tert-butoxycarbonyl-2-[2-methoxycarbonyl-(E)-ethenyl]-aziridine 
• 13734-34-4 N-tert-butoxycarbonyl-L-phenylalanine 
• 87694-53-9 Boc-Phe-OH N,O-dimethyl hydroxamate 
• 134210-25-6 (4R,5S)-5-[(tert-butoxycarbonyl)amino]-4-hydroxy-6-phenyl-(E)-2-hexenoate 
• 124266-92-8 Methyl (3R,4R,5S)-5-<(tert-butoxycarbonyl)amino>-3,4-epoxy-6-phenylhexanoate 
• 178259-04-6 methyl (5S)-5-[N-(tert-butoxycarbonyl)amino]-4-oxo-6-phenyl-(E)-2-hexenoate 
• 256463-34-0 (S)-5-[(tert-butoxycarbonyl)amino]-1-hydroxy-6-phenyl-(E)-2-hexen-4-one 
• 160002-06-2 (S)-tert-butyl 3-oxo-1-phenylhex-5-en-2-ylcarbamate 
• 82042-48-6 (S)-5-<(tert-Butoxycarbonyl)amino>-6-phenyl-(E)-3-hexenoic acid 
• 118457-05-9 Methyl (S)-5-<(tert-butoxycarbonyl)amino>-6-phenyl-(E)-3-hexenoate 

Relevant academic research and scientific papers

Synthesis of a complete series of C-4 fluorinated Phe-Gly mimetics

The complete series of Boc-protected allylic mono- and difluorinated Phe-Gly methyl ester derivatives has been synthesized using facile methods. Diastereomeric allylic alcohol derivatives were used as key intermediates, cis- And trans-aziridine derivative

Novel L-Phe-Gly mimetics

The syntheses of some novel dipeptidomimetics of potential biological interest are described. The reactions started from the vinyl isostere of Phe-Gly and were performed in high yields. Stereochemically pure products were isolated.