256463-34-0

Upstream product

• 160002-06-2 (S)-tert-butyl 3-oxo-1-phenylhex-5-en-2-ylcarbamate 
• 87694-53-9 Boc-Phe-OH N,O-dimethyl hydroxamate 
• 13734-34-4 N-tert-butoxycarbonyl-L-phenylalanine 

Downstream Products

• 256463-40-8 methyl (5S)-5-[(tert-butoxycarbonyl)amino]-4,4-difluoro-6-phenyl-hexanoate 
• 256463-35-1 methyl (4S,5S)-5-[(tert-butoxycarbonyl)amino]-4-fluoro-6-phenyl-(E)-2-hexenoate 
• 178259-04-6 methyl (5S)-5-[N-(tert-butoxycarbonyl)amino]-4-oxo-6-phenyl-(E)-2-hexenoate 
• 256463-36-2 methyl (2S,3S)-3-benzyl-1-tert-butoxycarbonyl-2-[2-methoxycarbonyl-(E)-ethenyl]-aziridine 
• 144075-71-8 methyl (2R,3S)-3-benzyl-1-tert-butoxycarbonyl-2-(2-methoxycarbonyl-(E)-ethenyl)-aziridine 
• 144075-70-7 methyl (4R,5S)-5-[(tert-butoxycarbonyl)amino]-4-fluoro-6-phenyl-(E)-2-hexenoate 
• 134210-24-5 methyl (4S,5S,2E)-5-amino-N-<(tert-butyloxy)carbonyl>-4-hydroxy-6-phenyl-2-hexanoate 
• 134210-25-6 (4R,5S)-5-[(tert-butoxycarbonyl)amino]-4-hydroxy-6-phenyl-(E)-2-hexenoate 
• 135130-98-2 (4R)-4-{1-[(S)-(tert-butoxycarbonyl)amino]-2-phenylethyl}-γ-butyrolactone 
• 127445-58-3 methyl (5S)-5-[(tert-butoxycarbonyl)amino]-4-oxo-6-phenyl-hexanoate 

Relevant academic research and scientific papers

Synthesis of a complete series of C-4 fluorinated Phe-Gly mimetics

The complete series of Boc-protected allylic mono- and difluorinated Phe-Gly methyl ester derivatives has been synthesized using facile methods. Diastereomeric allylic alcohol derivatives were used as key intermediates, cis- And trans-aziridine derivative