146564-05-8Relevant articles and documents
Convenient synthesis of 4-alkyl, alkenyl, and alkynyl substituted N-(phenylsulfonyl)indoles
Ishibashi,Akamatsu,Iriyama,Ikeda
, p. 2150 - 2153 (2007/10/02)
The indolone 1 reacted with organomagnesium or lithium reagents to give the carbinols 6 and 10, which, upon treatment under appropriate acidic conditions or neutral thermal conditions, gave the 1-phenylsulfonylindoles 8 and 11 bearing various kinds of alk
A new, general entry to 4-substituted indoles. Synthesis of (S)-(-)-pindolol and (±)-chuangxinmycin
Ishibashi, Hiroyuki,Tabata, Takashi,Hanaoka, Kyoko,Iriyama, Hiroko,Akamatsu, Susumu,Ikeda, Masazumi
, p. 489 - 492 (2007/10/02)
A new method for synthesis of 4-substituted indoles has been developed by using the 7-arylthio-6-7-dihydroindol-4(5H) one 5 as a common intermediate. The method was applied to the synthesis of (S)-(-)-pindolol (11) and (±)-chuangxinmycin (16).