1465783-87-2Relevant academic research and scientific papers
Carbon-14 labeling of K777·HCl, a therapeutic agent for Chagas disease
Rhee, Sung-Whi,Bradford, Wallace W.,Malerich, Jeremiah P.,Tanga, Mary J.
, p. 461 - 463 (2014/03/21)
The antitrypanosomal agent K777·HCl was labeled with carbon-14 to support absorption, distribution, metabolism, and excretion studies of this potential new drug for the treatment of Chagas disease. The radiolabeled compound was prepared in eight steps from [14C(U)]-(L)-phenylalanine with a specific activity of 54.4 mCi/mmol and an overall radiochemical yield of 4.1%. Copyright
