147372-85-8Relevant academic research and scientific papers
SPIROCHROMANE DERIVATIVES
-
Page/Page column 37; 44, (2020/02/06)
The invention relates to spirochromane derivatives, or pharmaceutically acceptable salts, biologically active metabolites, pro-drugs, racemates, enantiomers, diastereomers, solvates and hydrates thereof, as well as to pharmaceutical compositions containin
CHROMAN - SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS
-
Page/Page column 140, (2012/09/10)
The invention relates to chroman spirocyclic piperidine amide derivatives useful as inhibitors of ion channels. The invention also provides pharmaceutically acceptable compositions comprising the compounds of the invention and methods of using the compositions in the treatment of various disorders.
Potent 3-spiropiperidine growth hormone secretagogues
Yang, Lihu,Morriello, Greg,Prendergast, Kristine,Cheng, Kang,Jacks, Tom,Chan, Wanda W.-S.,Schleim, Klaus D.,Smith, Roy G.,Patchett, Arthur A.
, p. 107 - 112 (2007/10/03)
Systematic SAR studies of the different regioisomers and homologues of the spiro(indane-1,4'-piperidine) moiety in the growth hormone secretagogue L-162,752 are presented. Among them, spiro(3H-1-benzopyran-2,3'-piperidine) was found to afford secretagogue
Substituted piperidinylpropanols
-
, (2008/06/13)
Compounds having the formula STR1 and the pharmaceutically acceptable salts thereof, wherein n is 0, 1 or 2; R1 is alkanoyl; and R2 is STR2 R3 is alkyl; R4 is cyano or hydroxy; R5 is hydroxy or alkano
