148869-73-2Relevant academic research and scientific papers
Studies on aromatase inhibitors. I. Synthesis and biological evaluation of 4-amino-4H-1,2,4-triazole derivatives
Okada, Minoru,Yoden, Toru,Kawaminami, Eiji,Shimada, Yoshiaki,Kudoh, Masafumi,Isomura, Yasuo,Shikama, Hisataka,Fujikura, Takashi
, p. 1871 - 1879 (2007/10/03)
Various 4-N-substituted amino-4H-1,2,4-triazole derivatives were synthesized and evaluated for aromatase-inhibitory activity (in vitro) and for pregnant mare serum gonadotropin (PMSG)-induced estrogen synthesis- inhibitory activity (in vivo). The 4-(4-cya
