150555-92-3Relevant academic research and scientific papers
Metal-free visible light-promoted synthesis of isothiazoles: A catalytic approach for N-S bond formation from iminyl radicals under batch and flow conditions
Alemán, José,Berton, Mateo,Cabrera-Afonso, María Jesús,Cembellín, Sara,Halima-Salem, Adnane,Maestro, M. Carmen,Marzo, Leyre,Miloudi, Abdellah
supporting information, p. 6792 - 6797 (2020/11/09)
A sustainable synthesis of isothiazoles has been developed using an α-amino-oxy acid auxiliary and applying photoredox catalysis. This simple strategy features mild conditions, broad scope and wide functional group tolerance representing a new enviromenta
DIARYLSULFONES AS 5-HT2A ANTAGONISTS
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Page/Page column 27, (2008/06/13)
Compounds of formula (I) are potent and selective antagonists of the human 5-HT2A receptor, and hence useful in treatment of a variety of adverse conditions of the CNS.
Preparation of 6-fluorobenzisothiazoles via a regioselective nucleophilic aromatic substitution reaction
Fink,Strupczewski
, p. 6525 - 6528 (2007/10/02)
An efficient three step procedure for the preparation of 6-fluoro-1,2-benzisothiazoles is described. The key step is a regioselective nucleophilic aromatic substitution reaction in which the carbonyl group of a ketone or aldehyde directs nucleophilic disp
A method and intermediates for the preparation of 6-fluorobenzisothiazoles
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, (2008/06/13)
A process for the preparation of 6-fluoro-1,2-benzisothiazoles of formula I where R is hydrogen, loweralkyl, cycloalkyl, aralkyl, aryl, or a group of the formulae -CO2R2, -CN or -C(=O)R;2 R2 is alkyl or aryl; k,
