153546-07-7Relevant articles and documents
Asymmetric synthesis of photophore-containing lactisole derivatives to elucidate sweet taste receptors
Hashimoto, Makoto,Ishida, Akiko,Misaka, Takumi,Nakagita, Tomoya,Tachrim, Zetryana Puteri,Wang, Lei
, (2020/06/30)
Lactisole, which has a 2-phenoxy propionic acid skeleton, is well-known as an inhibitor of sweet taste receptors. We recently revealed some of the structure-activity relationships of the aromatic ring and chiral center of lactisole. Photoaffinity labeling
PIPERIDINE DERIVATES FOR THE TREATMENT OF CHEMOKINES MEDIARED DISEASE
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Page/Page column 29-30, (2010/02/14)
The present invention provides a compound of a formula (I) wherein the variables are defined herein; to a process for preparing such a compound; and to the use of such a compound in the treatment of a chemokine (such as CCR3) or H1 mediated disease state.