156604-31-8Relevant academic research and scientific papers
BACTERIAL EFFLUX PUMP INHIBITORS
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Page/Page column 40, (2017/09/09)
Disclosed herein are compounds of formula I: and salts thereof. Also disclosed are compositions comprising compounds of formula I and methods using compounds of formula I.
New analogues of agmatine with higher affinity to imidazoline receptors
Treder, Adam P.,Andruszkiewicz, Ryszard,Zgoda, W?odzimierz,Ford, Celeste,Hudson, Alan L.
scheme or table, p. 1009 - 1011 (2009/09/25)
Compilation of agmatine structure and imidazoline ring leads to a new family of imidazoline/α2-adrenoceptor ligands, 4(5)-(2-aminoethyl)imidazoline derivatives. Constraining of the guanidine moiety into heterocyclic ring improved the affinities of the resultant fusion compounds in comparison to agmatine itself. In this work, the synthetic approach and results for I1, I2, and α2-adrenoceptors affinities are reported.
A new approach to the synthesis of selectively protected (2S)-1,2,4-triaminobutane derivatives
Treder, Adam P.,Walkowiak, Aleksandra,Zgoda, Wlodzimierz,Andruszkiewicz, Ryszard
, p. 2281 - 2283 (2007/10/03)
An efficient synthesis of selectively protected (2S)-1,2,4-triaminobutane from L-glutamic acid via (2S)-N4-benzyloxycarbonyl-2,4- diaminobutanamid is described. Georg Thieme Verlag Stuttgart.
Selectively Protected Chiral 1,2,4-Triaminobutanes and Chiral Vicinal 1,2-Diamines
Altman, Janina,Ben-Ishai, Dov,Beck, Wolfgang
, p. 887 - 894 (2007/10/02)
Stepwise t-butoxycarbonylation of (S)-5-aminomethyl-2-pyrrolidone to mono-, di- and triacylated compounds has been elaborated.Ring opening of (S)-5-(Boc-aminomethyl)-N1-Boc-2-pyrrolidone with LiOH afforded the Boc-protected 4,5-diaminovaleric a
