1620108-59-9

Upstream product

• 53595-65-6 5-bromo-thiophene-2-sulfonamide 
• 209919-30-2 4-chloro-2-methylphenylboronic acid 
• 1620108-43-1 C₇H₆BClF₃^(1-)*K⁽¹⁺⁾ 

Relevant academic research and scientific papers

DIPHENYL SUBSTITUTED THIOPHENE-2-AMIDE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF USEFUL AS ANTIMICROBIAL

Compounds or pharmaceutical acceptable salts thereof of Formula (I), in which RM have the meaning described herein and pharmaceutical compositions thereof useful as antimicrobial and/or adjuvant:

Arylation and heteroarylation of thienylsulfonamides with organotrifluoroborates

A mild, practical protocol has been developed for the Suzuki cross-coupling of unprotected thienylsulfonamides from air- and bench-stable organotrifluoroborates in the absence of a protecting group on the sulfonamide nitrogen. The developed synthetic method can be applied to the preparation of various arylated and heteroarylated thienylsulfonamides under conditions that are tolerant of a broad range of functional groups.