164713-49-9Relevant academic research and scientific papers
Catalytic asymmetric diazoacetate cyclopropanation of 1-tosyl-3- vinylindoles. A route to conformationally restricted homotryptamines
Marcin, Lawrence R.,Denhart, Derek J.,Mattson, Ronald J.
, p. 2651 - 2654 (2007/10/03)
(Chemical Equation Presented) Substituted 1-tosyl-3-vinylindoles undergo catalytic asymmetric cyclopropanation with ethyl- and tert-butyldiazoacetate to afford N-protected trans-2-(indol-3-yl)-1-cyclopropanecarboxylic esters in good yield and high enantio
Stereoselective Synthesis of trans-2-(Indol-3-yl)cyclopropylamines: Rigid Tryptamine Analogues
Vangveravong, Suwanna,Nichols, David E.
, p. 3409 - 3413 (2007/10/02)
A procedure for the preparation of trans-2-(indol-3-yl)cyclopropylamines is reported.The key step in the sequence is a stereoselective palladium-catalyzed cyclopropanation of the indole-3-acryloyl derivative of Oppolzer's chiral sultam (bornanesulta
