179622-66-3Relevant academic research and scientific papers
Discovery of the first non-peptide full agonists for the human bradykinin B2 receptor incorporating 4-(2-picolyloxy)quinoline and 1-(2-picolyl)benzimidazole frameworks
Sawada, Yuki,Kayakiri, Hiroshi,Abe, Yoshito,Mizutani, Tsuyoshi,Inamura, Noriaki,Asano, Masayuki,Hatori, Chie,Aramori, Ichiro,Oku, Teruo,Tanaka, Hirokazu
, p. 2853 - 2863 (2007/10/03)
In the course of our studies on non-peptide bradykinin (BK) B2 receptor ligands, it was suggested that the 4-substituent of the quinoline ring may play a critical role in determining binding affinities for human and guinea pig B2 rec
Pyridopyrimidones, quinolines and fused N-heterocycles as bradykinin antagonists
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, (2008/06/13)
This invention relates to a compound of the formula: STR1 wherein Z is a group of the formula: STR2 in which X1 is N or C--R1, X2 is N or C--R9, X3 is N or C--R2, R1 is lower alk
