19195-31-4Relevant academic research and scientific papers
Bioglycerol-based sulfonic acid-functionalized carbon catalyst as an efficient and reusable catalyst for one-pot synthesis of 3- substituted-2 h -1,4-benzothiazines
Yang, Xiaojuan,Wu, Liqiang
, p. 1327 - 1333 (2013/10/08)
A simple and efficient synthetic protocol has been developed for the synthesis of 3-substituted-2H-1,4-benzothiazines by using bioglycerol-based sulfonic acid-functionalized carbon catalyst, devoid of corrosive acidic and basic reagents. The developed met
[Ir(P-OP)]-catalyzed asymmetric hydrogenation of diversely substituted C=N-containing heterocycles
Nunez-Rico, Jose Luis,Vidal-Ferran, Anton
supporting information, p. 2066 - 2069 (2013/06/04)
Iridium(I) complexes of enantiomerically pure phosphine-phosphite ligands ([Ir(Cl)(cod)(P - OP)]) efficiently catalyze the enantioselective hydrogenation of diverse C=N-containing heterocyclic compounds (benzoxazines, benzoxazinones, benzothiazinones, and quinoxalinones; 25 examples, up to 99% ee). A substrate-to-catalyst ratio as high as 2000:1 was reached.
Practical and efficient synthesis of 3-aryl-2H-benzo[1,4]thiazine derivatives catalyzed by KHSO4
Baghernejad, Bita,Heravi, Majid M.,Oskooie, Hossein A.
experimental part, p. 589 - 593 (2011/04/15)
KHSO4 efficiently catalyzes the condensation of o-aminothiophenols and 2-bromo-1-aryl-ethanones to yield 3-aryl-2H-benzo[1,4] thiazines in good yields.
From phenothiazine to 3-phenyl-1,4-benzothiazine derivatives as inhibitors of the Staphylococcus aureus NorA multidrug efflux pump
Sabatini, Stefano,Kaatz, Glenn W.,Rossolini, Gian Maria,Brandini, David,Fravolini, Arnaldo
experimental part, p. 4321 - 4330 (2009/05/07)
Overexpression of efflux pumps is an important mechanism by which bacteria evade effects of substrate antimicrobial agents and inhibition of such pumps is a promising strategy to circumvent this resistance mechanism. NorA is a Staphylococcus aureus multid
Conversion of bis(o-nitrophenyl)disulfides to heterocycles containing sulfur and nitrogen by the action of samarium diiodide
Zhong, Weihui,Chen, Xiaoyuan,Zhang, Yongmin
, p. 156 - 160 (2007/10/03)
Treatment of bis(o-nitrophenyl)disulfides 1 with SmI2 led to simultaneous reduction of nitro groups and reductive cleavage of S-S bonds as well as the formation of the active intermediates 2. The intermediates 2 reacted smoothly with aldehydes
New dyes based on 3-aryl-benzo- and -naphtho-1,4-thiazines
MacKenzie, Neil E.,Thomson, Ronald H.,Greenhalgh, Colin W.
, p. 2923 - 2932 (2007/10/02)
3-Aryl-2H-1,4-benzothiazines have been converted into cyanine dyes by condensing their hydroperchlorates with aldehydes, and into azo-compounds by coupling with reactive diazonium salts. The azo-compounds were also obtained by condensing arylglyoxal hydra
