19832-75-8Relevant academic research and scientific papers
I2-Promoted Intramolecular Oxidative Cyclization of Butenyl Anilines: A Facile Route to Benzo[b]azepines
An, Zhenyu,Ren, Yi,Liu, Yafeng,Yan, Rulong
, p. 2614 - 2617 (2021/08/06)
A metal-free approach for the synthesis of seven-membered N-heterocycles has been developed by the I2-promoted intramolecular cross-coupling/annulation of butenyl anilines. This cyclization reaction involves C?H activation and C?C bond formation and exhibits good functional group tolerance. A series of benzo[b]azepine derivatives are obtained in moderate to good yields.
Construction of N-Alkyl- and N-Arylaziridines from Unprotected Amines via C-H Oxidative Amination Strategy
Yu, Yang,Li, Meijuan,Zhang, Yong,Liu, Yonghai,Shi, Lei,Wang, Wei,Li, Hao
supporting information, p. 904 - 907 (2019/05/16)
A copper-promoted intramolecular C-H oxidative amination reaction between secondary amine (N-H) and C(sp3)-H at the benzylic position of azaarenes or α-position of ketones for the synthesis of aziridine derivatives has been developed. Moreover,
Synthesis of Heterocyclic Compounds: Part XXVIII - Potential Antileukemic Agents from 3,4-Dihydro-1,3,2-oxazaphosphorin-2-oxides
Sahasrabudhe, S. D.,Tilak, B. D.
, p. 914 - 917 (2007/10/02)
Some 3,6-diaryl-2-chloro-3,4-dihydro-1,3,2-oxazaphosphorin-2-oxides (4a-q, 6a-e and 7a, b) have been synthesised and tested for their anti-leukemic activity.
