219910-64-2Relevant academic research and scientific papers
Functionalization at position 3 of the phenyl ring of the potent mGluR5 noncompetitive antagonists MPEP
Alagille, David,Baldwin, Ronald M.,Roth, Bryan L.,Wroblewski, Jarda T.,Grajkowska, Ewa,Tamagnan, Gilles D.
, p. 945 - 949 (2005)
We described the synthesis and biological evaluation of MPEP analogs functionalized at the position 3 of the phenyl ring. The results point out the limitation in the choice of a functional group at this position; the only substituents leading to retention
Pyridine derivatives
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Page column 11, (2008/06/13)
A compound of formula I wherein X represents an optionally halo-substituted (C2-4)alkynylene group bonded via vicinal unsaturated carbon atoms.
