2513-76-0Relevant academic research and scientific papers
Microbial transformation of parthenolide
Galal, Ahmed M.,Ibrahim, Abdel-Rahim S.,Mossa, Jaber S.,El-Feraly, Farouk S.
, p. 761 - 765 (1999)
Microbial transformation of the germacranolide parthenolide using Rhizopus nigricans, Streptomyces fulvissimus and Rhodotorula rubra yielded three new compounds: 11αH-dihydroparthenolide, 9β-hydroxy-11βH- dihydroparthenolide and 14-hydroxy-11βH-dihydroparthenolide. 11βH- dihydroparthenolide was the only common metabolite produced by all microorganisms.
Aminoparthenolides as novel anti-leukemic agents: Discovery of the NF-κB inhibitor, DMAPT (LC-1)
Neelakantan, Sundar,Nasim, Shama,Guzman, Monica L.,Jordan, Craig T.,Crooks, Peter A.
body text, p. 4346 - 4349 (2010/04/05)
A series of aminoparthenolide analogs (6-37) were synthesized and evaluated for their anti-leukemic activity. Eight compounds exhibited good anti-leukemic activity with LD50's in the low μM range (1.5-3.0 μM). Compounds 16, 24 and 30 were the m
