2836-44-4Relevant academic research and scientific papers
Novel pyrimidine derivatives containing an amide moiety: design, synthesis, and antifungal activity
Wu, Wenneng,Chen, Meihang,Wang, Rui,Tu, Haitang,Yang, Maofa,Ouyang, Guiping
, p. 719 - 729 (2019)
The objectives of the current study were to synthesize a series of novel pyrimidine derivatives containing an amide moiety and to investigate their in vitro antifungal activities against eight kinds of plant pathogenic fungi via the poison plate technique
Synthesis and Antifungal and Insecticidal Activities of Novel N -Phenylbenzamide Derivatives Bearing a Trifluoromethylpyrimidine Moiety
Yu, Xuetong,Lan, Wenjun,Chen, Meihang,Xu, Su,Luo, Xiaoxi,He, Shuhong,Chen, Haijiang,Fei, Qiang,Wu, Wenneng
, (2021/10/07)
Seventeen novel N-phenylbenzamide derivatives bearing a trifluoromethylpyrimidine moiety were synthesized via four-step reactions. Their antifungal and insecticidal properties were evaluated. Antifungal test results demonstrated that some of the synthesized compounds showed better in vitro bioactivities against Phomopsis sp., Botryosphaeria dothidea (B. dothidea), and Botrytis cinerea (B. cinerea) at 50 μg/mL than pyrimethanil. Unfortunately, the synthesized compounds revealed lower insecticidal activities against Spodoptera frugiperda (S. frugiperda) and Mythimna separata (M. separata) at 500 μg/mL than chlorantraniliprole.
Trifluoromethyl pyrimidine containing Ferulamide derivative and preparation and use thereof
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Paragraph 0020; 0022-0023, (2019/08/20)
The invention discloses a trifluoromethyl pyrimidine containing Ferulamide derivative. The trifluoromethyl pyrimidine containing Ferulamide derivative is characterized by having a structural general formula represented by (I) shown in the description, wherein R1 is H, methyl, ethyl, n-propyl, isopropyl, n-butyl, phenyl, methylmercapto, ethylmercapto, fluoro-, chloro-, bromo-, trifluoromethyl and N,N-dimethylamine, R2 is monosubstituted, disubstituted and trisubstituted, and R2 is H, methyl, ethyl, methoxy, ethoxy, fluoro-, chloro-, bromo-, iodo-, trifluoromethyl, nitro- and hydroxyl. The trifluoromethyl pyrimidine containing Ferulamide derivative can resist major pathogenic bacteria, i.e., Phomopsis Sp. and Botryosphaeria dothidea of kiwi fruit soft rot.
PYRIMIDINE COMPOUND AND ITS USE IN PEST CONTROL
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Page/Page column 175; 176, (2010/12/18)
A pyrimidine compound represented by below formula (I) has excellent control activity against pests and is useful as an active ingredient of a pest controlling agent.
PYRIMIDINE DERIVATIVES AND HERBICIDES CONTAINING THE SAME
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, (2008/06/13)
The present invention provides a pyrimidine derivative represented by the formula: wherein R1p and R1q are the same or different, and each represents (1)hydrogen, (2)halogen, (3) a C1-6alkyl group which may be substituted or (4) a C1-6alkoxy group, and so on, R2 is halogen, a C1-6alkyl group, cyano group, and so on, Ar is a phenyl group which may be substituted or is a condensed hetero ring which may be substituted, which has excellent selective herbicidal activity, and a herbicide containing the derivative.
