284465-88-9Relevant academic research and scientific papers
Facile synthesis of 3-arylpyrroles by tandem Suzuki-dehydrogenation reaction
Lee, Chi-Wan,Chung, Yong Jun
, p. 3423 - 3425 (2000)
Facile method for the synthesis of 3-arylpyrroles is described based on the palladium-catalyzed coupling of trifluoromethanesulfonic acid 1-benzyl- 2,5-dihydro-1H-pyrrol-3-yl ester with aryl halides. (C) 2000 Elsevier Science Ltd.
SUBSTITUTED OXETANES AND THEIR USE AS INHIBITORS OF CATHEPSIN C
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Page/Page column 50; 51, (2016/03/04)
This invention relates to a compound of formula I and their use as inhibitors of Cathepsin C, pharmaceutical compositions containing the same, and methods of using the same as agents for treatment and/or prevention of diseases connected with dipeptidyl peptidase I activity, e.g. respiratory diseases.
SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C
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Page/Page column 228-229, (2014/09/29)
This invention relates to 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)- amides of formula (1) and their use as inhibitors of Cathepsin C, pharmaceutical compositions containing the same, and methods of using the same as agents for treatment and/or prevention of diseases connected with dipeptidyl peptidase I activity, e.g. respiratory diseases.
SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C
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Paragraph 0604 - 0607; 0610, (2014/09/29)
This invention relates to 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid(benzyl-cyano-methyl)-amides of formula 1 and their use as inhibitors of Cathepsin C, pharmaceutical compositions containing the same, and methods of using the same as agents for treatment and/or prevention of diseases connected with dipeptidyl peptidase I activity, e.g. respiratory diseases.
