328546-89-0Relevant articles and documents
Tricyclic benzimidazoles as potent poly(ADP-ribose) polymerase-1 inhibitors
Skalitzky, Donald J.,Marakovits, Joseph T.,Maegley, Karen A.,Ekker, Anne,Yu, Xiao-Hong,Hostomsky, Zdenek,Webber, Stephen E.,Eastman, Brian W.,Almassy, Robert,Li, Jianke,Curtin, Nicola J.,Newell, David R.,Calvert, A. Hilary,Griffin, Roger J.,Golding, Bernard T.
, p. 210 - 213 (2007/10/03)
Novel tricyclic benzimidazole carboxamide poly-(ADP-ribose) polymerase-1 (PARP-1) inhibitors have been synthesized. Several compounds were found to be powerful chemopotentiators of temozolomide and topotecan in both A549 and LoVo cell lines. In vitro inhi