3327-79-5Relevant academic research and scientific papers
MORPHAN AND MORPHINAN ANALOGUES, AND METHODS OF USE
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Page/Page column 74, (2014/12/12)
The present application relates to analogues of morphan and morphinan, compositions thereof, and methods for treating a disease or condition comprising administering an effective amount of the compounds or compositions to a subject in need thereof.
Synthesis and pharmacological evaluation of 6,7-indolo/thiazolo-morphinans - Further SAR of levorphanol
Zhang, Ao,Li, Fuying,Ding, Chunyong,Yao, Qizhen,Knapp, Brian I.,Bidlack, Jean M.,Neumeyer, John L.
, p. 2747 - 2751 (2008/02/07)
To further extend the structure-activity relationships of levorphanol, two series of novel morphinans were prepared by incorporation of an indole or aminothiazole fragment to the hexyl ring (ring C) in levorphanol. Such morphinans differed from previously reported ligands in that such indole- or aminothiazole-containing morphinans displayed enhanced binding affinity to the δ opioid receptor, while the affinity to κ and μ receptors was slightly reduced.
