333350-50-8Relevant academic research and scientific papers
Copper-catalyzed amide bond formation from formamides and carboxylic acids
Liu, Hong-Qiang,Liu, Jun,Zhang, Yang-Hui,Shao, Chang-Dong,Yu, Jing-Xun
, p. 11 - 14 (2015/01/30)
A highly efficient copper-catalyzed approach to form amide bonds from formamides and carboxylic acids was developed. This protocol shows broad substrate scopes and high yields in the presence of 1 mol% catalyst and 4.0 equiv. formamides.
Therapeutically Active Thiazolo-Pyrimidine Derivatives
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Paragraph 0249, (2014/10/29)
A series of thiazolo[5,4-d]pyrimidine derivatives of formula (I) or an N-oxide thereof, or a pharmaceutically acceptable salt or solvate thereof: (I) Q represents a group of formula (Qa), (Qb), (Qc), (Qd) or (Qe) are beneficial in the treatment and/or prevention of various human ailments, including inflammatory, autoimmune and oncological disorders; viral diseases; and organ and cell transplant rejection.
THERAPEUTICALLY ACTIVE THIAZOLO-PYRIMIDINE DERIVATIVES
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Page/Page column 47, (2013/05/23)
A series of thiazolo[5,4-d]pyrimidine derivatives of formula (I) or an N-oxide thereof, or a pharmaceutically acceptable salt or solvate thereof: (I) Q represents a group of formula (Qa), (Qb), (Qc), (Qd) or (Qe) are beneficial in the treatment and/or prevention of various human ailments, including inflammatory, autoimmune and oncological disorders; viral diseases; and organ and cell transplant rejection.
Tetrahydropteridines useful as inhibitors of protein kinases
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Page/Page column 23, (2009/04/24)
The present invention relates to compounds useful as inhibitors of protein kinase. The invention also provides pharmaceutically acceptable compositions comprising said compounds and methods of using the compositions in the treatment of various disease, co
A rapid synthesis of 2-aryl-5-substituted-2,3-dihydrobenzofurans
Kuethe, Jeffrey T.,Wong, Audrey,Journet, Michel,Davies, Ian W.
, p. 3727 - 3729 (2007/10/03)
(Chemical Equation Presented) An effective strategy has been developed for the rapid and efficient one-pot synthesis of 2-aryl-5-substituted-2,3- dihydrobenzofurans from readily available o-nitrotoluenes and aromatic aldehydes. This strategy allows access to a structurally diverse array of products for further manipulation.
