342613-80-3Relevant academic research and scientific papers
ISOQUINOLINE DERIVATIVES AS PROTEIN KINASE INHIBITORS
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Page/Page column 199, (2021/02/12)
The present invention relates to a compound suitable for use as a kinase inhibitor
AMIDE COMPOUNDS, COMPOSITIONS AND USES THEREOF
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Page/Page column 64, (2009/10/22)
Compounds are provided according to formula (1 ) : where A, B, W, X', L, R1, R3, R4b, and m' are as defined herein. Provided compounds and pharmaceutical compositions thereof are useful for the prevention and treatment of a variety of conditions in mammals including humans, including by way of non-limiting example, pain, inflammation, cognitive disorders, anxiety, depression, and others.
IMIDAZOPYRIDINE DERIVATIVES AS INHIBITORS OF RECEPTOR TYROSINE KINASES
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Page/Page column 116, (2010/01/07)
The invention relates to new bicyclic heterocyclic derivative compounds, to pharmaceutical compositions comprising said compounds and to the use of said compounds in the treatment of diseases, e.g. cancer.
PIPERIDINE DERIVATIVES USEFUL AS HISTAMINE H3 ANTAGONISTS
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Page/Page column 51, (2010/11/25)
Disclosed are novel compounds of the formula (I) or a pharmaceutically acceptable salt thereof, wherein: M1 and M3 are CH or N; M2 is CH, CF or N; Y is -C(=O)-, -C(=S)-, -(CH2)q-, -C(=NOR7)
Heterocyclization of functionalized vinylic derivatives of imidazo[1,2-α]pyridines
Chezal,Moreau,Delmas,Gueiffier,Blache,Grassy,Lartigue,Chavignon,Teulade
, p. 6576 - 6584 (2007/10/03)
Heterocyclization of functionalized vinylic derivatives of imidazo[1,2-α]pyridines was explored experimentally and theoretically using semiempirical AM1 and ab initio methods. A range of functionalized vinylic derivatives (azido, amino, and carbodiimide groups) were prepared for conversion into pyrroloazaindoles 19-22, imidazo[1,x]-; (x=5, 6, 7, 8), [2,6]-, and [2,7]naphthyridines 28-30, 35-38 by thermal reaction. In the case of vinylic groups in the 5 position, peri annulation also was observed. The experimental and theoretical data are compared and discussed.
