449170-65-4Relevant articles and documents
Evaluation of diarylureas for activity against plasmodium falciparum
Zhang, Yiqun,Anderson, Marc,Weisman, Jennifer L.,Lu, Min,Choy, Cindy J.,Boyd, Vincent A.,Price, Jeanine,Sigal, Martina,Clark, Julie,Connelly, Michele,Zhu, Fangyi,Guiguemde, W. Armand,Jeffries, Cynthia,Yang, Lei,Lemoff, Andrew,Liou, Ally P.,Webb, Thomas R.,Derisi, Joseph L.,Guy, R. Kiplin
scheme or table, p. 460 - 465 (2011/02/27)
A library of diarylurea insulin-like growth factor 1 receptor inhibitors was screened for activity against chloroquine-sensitive (3D7) and chloroquine-resistant (K1) strains of Plasmodium falciparum. The 4-aminoquinaldine-derived diarylureas displayed pro