494221-67-9Relevant articles and documents
Discovery of an 8-aza-5-thiaProstaglandin E1 analog as a highly selective EP4 receptor agonist
Kambe, Tohru,Maruyama, Toru,Naganawa, Atsushi,Asada, Masaki,Seki, Akiteru,Maruyama, Takayuki,Nakai, Hisao,Toda, Masaaki
, p. 1494 - 1508 (2012/01/13)
For the purpose of discovering an orally available EP4 subtype-selective agonist, a series of 8-aza prostaglandin E1 (PGE1) analogs were synthesized and evaluated for their affinity for PGE2 receptor subtypes. Additionally