52459-55-9Relevant academic research and scientific papers
Synthesis and pharmacological characterisation of 2,4-dicarboxy-pyrroles as selective non-competitive mGluR1 antagonists.
Micheli, Fabrizio,Fabio, Romano Di,Cavanni, Paolo,Rimland, Joseph M,Capelli, Anna Maria,Chiamulera, Cristiano,Corsi, Mauro,Corti, Corrado,Donati, Daniele,Feriani, Aldo,Ferraguti, Francesco,Maffeis, Micaela,Missio, Andrea,Ratti, Emiliangelo,Paio, Alfredo,Pachera, Roberta,Quartaroli, Mauro,Reggiani, Angelo,Sabbatini, Fabio Maria,Trist, David G,Ugolini, Annarosa,Vitulli, Giovanni
, p. 171 - 183 (2007/10/03)
Metabotropic glutamate receptors (mGluRs) are an unusual family of G-protein coupled receptor (GPCR), and are characterised by a large extracellular N-terminal domain that contains the glutamate binding site. We have identified a new class of non-competit
