54127-64-9Relevant academic research and scientific papers
Pyridine phenyl coupling compound and pharmaceutical composition and application thereof
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Paragraph 0103; 0104; 0105, (2016/12/22)
The invention discloses a pyridine phenyl coupling compound and a pharmaceutical composition and application thereof. The pyridine phenyl coupling compound is a PSD-95-nNOs uncoupling agent, can selectively inhibit combination between PSD-95 and nNOs to a
New compounds, pharmaceutical compositions and uses thereof
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, (2012/09/05)
The invention relates to new compounds of the formula I to their use as medicaments, to methods for their therapeutic use and to pharmaceutical compositions containing them.
SEPIAPTERIN REDUCTASE INHIBITORS FOR THE TREATMENT OF PAIN
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Page/Page column 98-99, (2011/05/05)
Disclosed herein are small molecule heterocyclic inhibitors of sepiapterin reductase (SPR), and pro-drugs and pharmaceutically acceptable salts thereof. The Also featured are pharmaceutical compositions of the compounds and uses of these compounds for the treatment or prevention of pain (e.g., inflammatory pain, nociceptive pain, functional pain, and neuropathic pain)
3-PYRIDINYLETHYLBENZAMIDE DERIVATIVES AS FUNGICIDES
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Page/Page column 25, (2008/06/13)
Compound of general formula (I). Process for preparing this compound. Intermediate of general formula (II) to prepare compound of formula (I). Intermediate of general formula (V) to prepare compound of formula (I). Fungicidal composition comprising a comp
2-(3-Amino-2-hydroxy-propoxy)-mono-and diazines
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, (2008/06/13)
Heterocyclic compounds of the formula STR1 wherein Het denotes optionally substituted pyridazinyl, pyrimidinyl, pyrazinyl or substituted pyridyl, R1 is hydrogen or methyl and R2 is lower alklyl, optionally substituted phenyl-lower alkyl, carboxy-lower alkyl or functionally modified carboxy-lower alkyl, their condensation products with aldehydes, ketones or carbonic acid and their N-oxides, which are valuable (cardioselective) β-receptor blocking agents, and/or (cardioselective) β-receptor-stimulants.
2-(3-AMINO-2-HYDROXY-PROPOXY)-PYRAZINES
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, (2008/06/13)
Heterocyclic compounds of the formula STR1 wherein Het denotes optionally substituted pyridazinyl, pyrimidinyl, pyrazinyl or substituted pyridyl, R 1 is hydrogen or methyl and R 2 is lower alkyl, optionally substituted phenyl-lower alkyl, carboxy-lower alkyl or functionally modified carboxy-lower alkyl, their condensation products with aldehydes, ketones or carbonic acid and their N-oxides, which are valuable (cardioselective) β-rezeptor blocking agents, and/or (cardioselective) β-rezeptor-stimulants.
