57676-04-7Relevant articles and documents
Condensed 1,3-Benzothiazinones. 2. Synthesis of 2-Substituted 1,2,4-Triazolobenzothiazin-9-ones
Liu, Kang-Chien,Shih, Bi-Jane,Chern, Ji-Wang
, p. 457 - 460 (2007/10/02)
Heating 3-amino-2-imino-3,4-dihydro-2H-1,3-benzothiazin-4-one (1) with formic acid neat or with trimethyl orthoformate (2a) in xylene gave 1,2,4-triazolobenzothiazin-9-one (3a) in 49 and 81percent yields, respectively.An analogous reaction of
Cyanogen condensations as a route to 3 amino 2 imino 1,3 benzothiazin 4 ones with CNS depressant potential
Heindel,Schaeffer
, p. 1425 - 1427 (2007/10/05)
Seven new 3 amino 2 imino 1,3 benzothiazin 4 ones, prepared from the condensation of cyanogen and 2 mercaptobenzhydrazides, were evaluated in a neuropharmacological mouse profile. CNS depression was observed in several members of the class.