58668-52-3Relevant academic research and scientific papers
Design and synthesis of conformationally constraint Dyrk1A inhibitors by creating an intramolecular H-bond involving a benzothiazole core
Salah, Mohamed,Abdel-Halim, Mohammad,Engel, Matthias
, p. 1045 - 1053 (2018/06/27)
We present the development of conformationally pre-organised Dyrk1A inhibitors based on the hydroxybenzothiazole urea scaffold. The modifications introduced to the discovered hit (AHS-211) proved the crucial role of the urea linker to preserve the bioacti
N-(6-acyloxybenzothiazol-2-yl)-N'-phenyl (or substituted phenyl)ureas
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, (2008/06/13)
N-(6-Acyloxybenzimidazol-2-yl)-N'-phenyl (or substituted pehnyl)ureas are useful as immune regulants.
