60230-69-5Relevant academic research and scientific papers
Copper(I)-catalyzed tandem cyclization/condensation reaction to novel 4,5-dihydropyrazolo[1,5-a]quinolines and pyrazolo[1,5-a]indoles
Hang, Chenchen,Li, Qiulian,Zhu, Yongming,Katayama, Hajime
experimental part, p. 3318 - 3324 (2011/09/15)
A facile copper(I)-catalyzed tandem reaction for the synthesis of 4,5-dihydropyrazolo[1,5-a]quinolines and pyrazolo[1,5-a]indoles is reported here. High efficiency and good yields are displayed in this transformation under mild reaction conditions.
Intramolecular Reaction of the Hydrazonyl Group with Formyl and Oxo Groups: Preparation of Pyrazoloindoles and Related Pyrazolo Compounds
Shen, Jing-Kang,Katayama, Hajime,Takatsu, Noriyuki,Shiro, Itsuo
, p. 2087 - 2098 (2007/10/02)
Lewis acid-catalysed intramolecular nucleophilic attack of a hydrazonyl group onto aldehyde and ketone groups gives pyrazoles and dihydropyrazoles.Pyrazoloindoles and related pyrazolo compounds have also been prepared.
Preparation of Pyrazole and Pyrazoline Derivatives by Intramolecular Reaction of Hydrazones
Shen, Jing-Kang,Katayama, Hajime
, p. 451 - 452 (2007/10/02)
Pyrazole and pyrazoline derivatives are prepared by the intramolecular cyclization reaction of a hydrazonyl group with formyl or keto groups in the presence of a Lewis acid.
Synthesis and pregnancy terminating activity of pyrazolo[1,5-a]indoles and quinolines
Winters,Odasso,Conti,et al.
, p. 215 - 218 (2007/10/02)
In order to clarify the structural requirements for antifertility activity, series of 2-arylpyrazolo[1,5-a]indoles and 2-arylpyrazolo[1,5-a]-quinolines were prepared and tested in rats and hamsters. Their potencies were compared with those of the isomeric
2-Phenyl-pyrazolo-[1,5-a]quinoline compounds
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, (2008/06/13)
New heterocyclic compounds represented by the following formula: STR1 wherein: R and R1 are independently selected from hydrogen, hydroxy, (C1-4)alkyl, (C1-4)alkoxy, (C3-5)alkenyloxy, (C3-5)alkynyloxy
