614735-34-1

Upstream product

• 824-94-2 p-methoxybenzyl chloride 
• 68724-96-9 10-methyl-1,2,3,4,5,10-hexahydroazepino[3,4-b]indole-1,5-dione 
• 1477-50-5 Indole-2-carboxylic acid 
• 68724-95-8 3-[(1-methyl-1H-indole-2-carbonyl)amino]propionic acid ethyl ester 
• 68724-78-7 3-[(1H-indole-2-carbonyl)amino]propionic acid ethyl ester 
• 68724-80-1 3-{[(1-methyl)-1H-2-indolylcarbonyl]amino}propanoic acid 

Downstream Products

• 614735-63-6 4-bromo-2-(4-methoxybenzyl)-10-methyl-3,4-dihydro-2H,10H-azepino[3,4-b]indole-1,5-dione 
• 614735-35-2 4,4-dibromo-2-(4-methoxybenzyl)-10-methyl-3,4-dihydro-2H,10H-azepino[3,4-b]indole-1,5-dione 
• 614735-54-5 2-(4-methoxybenzyl)-10-methyl-4-(1-ethoxyvinyl)-2H,10H-azepino[3,4-b]indole-1,5-dione 
• 614735-52-3 2-(4-methoxybenzyl)-10-methyl-4-vinyl-2H,10H-azepino[3,4-b]indole-1,5-dione 
• 614735-37-4 4-bromo-2-(4-methoxybenzyl)-10-methyl-2H,10H-azepino[3,4-b]indole-1,5-dione 
• 794547-73-2 ethyl 4-allyl-2-(4-methoxybenzyl)-10-methyl-1,5-dioxo-1,2,3,4,5,10-hexahydroazepino[3,4-b]indole-4-carboxylate 
• 794547-84-5 4-allyl-4-(3-butenyl)-2-(4-methoxybenzyl)-10-methyl-3,4-dihydroazepino[3,4-b]indole-1,5(2H,10H)-1,5-dione 

Relevant academic research and scientific papers

Synthesis and reactivity of azepino[3,4-b]indol-5-yl trifluoromethanesulfonate

A convenient method for the synthesis of 5-substituted azepino[3,4- b]indol-1-ones 18 - 27 is described. This synthesis was based on palladium mediated cross-coupling reactions of the key intermediate azepino[3,4- b]indol-5-yl trifluoromethanesulfonates 3, obtained from the corresponding azepino[3,4-b]indole-1,5-dione 4. (C) 2000 Elsevier Science Ltd.