6336-34-1Relevant articles and documents
Design, synthesis and evaluation of potent and selective inhibitors of mono-(ADP-ribosyl)transferases PARP10 and PARP14
Holechek, Jacob,Lease, Robert,Thorsell, Ann-Gerd,Karlberg, Tobias,McCadden, Caitlin,Grant, Ryan,Keen, Abby,Callahan, Evan,Schüler, Herwig,Ferraris, Dana
, p. 2050 - 2054 (2018)
A series of diaryl ethers were designed and synthesized to discern the structure activity relationships against the two closely related mono-(ADP-ribosyl)transferases PARP10 and PARP14. Structure activity studies identified 8b as a sub-micromolar inhibito
An artificial receptor for the intermolecular and enantioselective formation of peptide sheets
Eblinger, Frank,Schneider, Hans-Joerg
, p. 2297 - 2298 (2007/10/03)
Peptide strands coupled at the C terminus to bis[p(aminomethyl)phenyl] ether allow in CHCl3 solution association of lipophilic N-protected peptides with hydrogen bonds in the mode of antiparallel β-sheets; the enantioselectivity observed with a phenylalanine derivative is characterized by a binding constant ratio of around 15.